SCHEMBL624902

SCHEMBL624902

CN(C)c1cccc(-c2cnc3sc(C(C)(N)C4CCNCC4)nn23)c1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FYN P06241 13/20 0.54
PIK3CA P42336 1/20 0.40
DCTPP1 Q9H773 1/20 0.38
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
PTK2 Q05397 1/20 0.36
PIM1 P11309 2/20 0.35
PIK3CD O00329 1/20 0.35
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624903 0.77 FYN (0.53) FYNPIK3CADCTPP1JAK2JAK3
SCHEMBL625540 0.71 FYN (0.68) FYN
SCHEMBL15603228 0.70 FYN (0.49) FYNDCTPP1
SCHEMBL1944343 0.70 FYN (1.00) FYNPIM1
SCHEMBL1947153 0.69 FYN (0.48) FYNDCTPP1
SCHEMBL623882 0.69 DYRK1A (0.46) FYNPIM1
SCHEMBL1946908 0.68 FYN (0.47) FYNDCTPP1
SCHEMBL1946916 0.68 FYN (0.75) FYNPIM1
SCHEMBL1944499 0.67 FYN (0.58) FYN
SCHEMBL1944077 0.67 FYN (0.71) FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed