SCHEMBL624903

SCHEMBL624903

CN(C)c1cccc(-c2cnc3sc(N(C)CC4CCNCC4)nn23)c1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FYN P06241 14/20 0.53
PIK3CA P42336 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
JAK2 O60674 1/20 0.37
JAK3 P52333 1/20 0.37
PTK2 Q05397 1/20 0.37
DCTPP1 Q9H773 1/20 0.37
PIM1 P11309 2/20 0.36
PIM2 Q9P1W9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624008 0.83 PIM1 (0.56) PIM1PIM2
SCHEMBL624433 0.82 FYN (0.47) FYNJAK2JAK3PTK2PIM1
SCHEMBL624904 0.81 F2RL3 (0.41) FYNJAK2JAK3PTK2PIM1
SCHEMBL624902 0.77 FYN (0.54) FYNPIK3CAGRIN1GRIN2BJAK2
SCHEMBL623806 0.76 FYN (0.54) FYNPIM1PIM2
SCHEMBL15603322 0.72 FYN (0.50) FYNDCTPP1
SCHEMBL623882 0.72 DYRK1A (0.46) FYNPIM1PIM2
SCHEMBL1946916 0.71 FYN (0.75) FYNPIM1
SCHEMBL1946370 0.71 FYN (0.49) FYN
SCHEMBL625540 0.70 FYN (0.68) FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed