SCHEMBL6249303

SCHEMBL6249303

COC(=O)/C(=C/CCc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CTSK P43235 4/20 0.42
CTSS P25774 4/20 0.42
AKT1 P31749 3/20 0.41
SIGMAR1 Q99720 3/20 0.40
ATM Q13315 1/20 0.40
IDO1 P14902 1/20 0.39
CTSL P07711 2/20 0.39
CTSB P07858 2/20 0.39
KLK5 Q9Y337 1/20 0.38
PPARA Q07869 2/20 0.38
PPARG P37231 1/20 0.38
SYK P43405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6249304 1.00 CA12 (0.43) CA12CA1CA7CA14CTSK
SCHEMBL3867978 0.88 NPC1 (0.42) CA1CTSKCTSSAKT1IDO1
SCHEMBL13906650 0.77 LMNA (0.44) CA12CA1CA7CA14
SCHEMBL8434086 0.76 CA12 (0.48) CA12CA1
SCHEMBL17844739 0.76 CA12 (0.47) CA12CA1CA7CA14CTSK
SCHEMBL17844742 0.76 CA12 (0.47) CA12CA1CA7CA14CTSK
SCHEMBL19562463 0.76 PPARA (0.37) CA12CA1CA7CA14CTSK
SCHEMBL31536313 0.76 SYK (0.41) CA12CA1CA7CA14CTSS
SCHEMBL8837533 0.75 CA12 (0.49) CA12CA1CA7CA14CTSK
SCHEMBL26831798 0.75 TDP1 (0.34) CA12CA1CA7CA14CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005044810-A1 GLYT2 MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2005-05-19 WO disclosed