SCHEMBL624978

SCHEMBL624978

N#Cc1cccc(-c2cnc3sc(NC4CC5(CCNCC5)C4)nn23)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FYN P06241 14/20 0.51
PIM1 P11309 1/20 0.44
HASPIN Q8TF76 1/20 0.38
PLAT P00750 1/20 0.38
NTRK1 P04629 1/20 0.38
NTRK3 Q16288 1/20 0.38
NTRK2 Q16620 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
AKT1 P31749 1/20 0.37
AKT2 P31751 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625548 0.84 FYN (0.52) FYNPIM1
SCHEMBL625540 0.84 FYN (0.68) FYNHASPIN
SCHEMBL625560 0.82 FYN (0.50) FYNPIM1
SCHEMBL624036 0.82 FYN (0.46) FYNPIM1HSD17B10
SCHEMBL624979 0.81 ADORA2A (0.38) PIM1PLATCYP1A2CYP2C19HSD17B10
SCHEMBL623851 0.77 FYN (0.61) FYNPIM1NTRK1NTRK3NTRK2
SCHEMBL626107 0.75 PIK3CA (0.48) FYNHASPIN
SCHEMBL2255599 0.71 FYN (0.53) FYNNTRK1NTRK3NTRK2
SCHEMBL1945052 0.70 FYN (0.65) FYNHASPIN
SCHEMBL624945 0.69 FYN (0.49) FYNPIM1HASPIN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed