SCHEMBL6250485

SCHEMBL6250485

C=CC(=O)N[C@@H](CC(C)C)C(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 7/20 0.48
POLB P06746 5/20 0.48
TDP1 Q9NUW8 4/20 0.48
MAPT P10636 9/20 0.45
KMT2A Q03164 7/20 0.45
MEN1 O00255 5/20 0.45
ALDH1A1 P00352 2/20 0.45
RECQL P46063 3/20 0.44
XBP1 P17861 1/20 0.44
GAA P10253 1/20 0.43
TSHR P16473 1/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
MAPK1 P28482 3/20 0.41
ATM Q13315 2/20 0.41
NOS3 P29474 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21368437 1.00 NPSR1 (0.48) NPSR1POLBTDP1MAPTKMT2A
SCHEMBL21368257 0.84 TSHR (0.41) NPSR1POLBTDP1ALDH1A1TSHR
SCHEMBL21367972 0.83 TAS1R3 (0.55) POLBTSHRTAS1R3TAS1R1NOS3
SCHEMBL29820642 0.83 TAS1R3 (0.55) POLBTSHRTAS1R3TAS1R1NOS3
SCHEMBL16964411 0.83 TSHR (0.40) NPSR1POLBTDP1MAPTKMT2A
SCHEMBL21368436 0.81 TSHR (0.46) POLBALDH1A1TSHRTAS1R3TAS1R1
SCHEMBL21368435 0.81 PPID (0.46) TSHRTAS1R3TAS1R1NOS3NOS1
SCHEMBL21675512 0.80 CTSK (0.61) NPSR1POLBTDP1MAPTKMT2A
SCHEMBL27513177 0.79 NPSR1 (0.51) NPSR1POLBTDP1MAPTKMT2A
SCHEMBL21368254 0.78 TSHR (0.50) NPSR1POLBTDP1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1560630-A2 7H-DIBENZO[B,G][1,5]DIOXOCIN-5-ONE DERIVATIVES AND USE THEREOF Bayer HealthCare AG (DE) 2005-08-10 EP disclosed
WO-2004039453-A2 7H-DIBENZO[B,G][1,5]DIOXOCIN-5-ONE DERIVATIVES AND USE THEREOF BAYER HEALTHCARE AG (DE) 2004-05-13 WO disclosed