SCHEMBL6251414

SCHEMBL6251414

CCN(CC)CCNC(=O)c1ccc2c(ccn2C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.54
ALDH1A1 P00352 2/20 0.54
SLC22A2 O15244 1/20 0.54
SLC22A1 O15245 1/20 0.54
TSHR P16473 1/20 0.54
ACHE P22303 1/20 0.54
MAPK1 P28482 1/20 0.54
CYP2C19 P33261 1/20 0.54
BLM P54132 2/20 0.53
PMP22 Q01453 1/20 0.53
TMEM97 Q5BJF2 1/20 0.52
SIGMAR1 Q99720 1/20 0.52
NFKB1 P19838 1/20 0.51
KCNH2 Q12809 1/20 0.51
HDAC3 O15379 1/20 0.51
HDAC1 Q13547 1/20 0.51
POLB P06746 2/20 0.50
CD274 Q9NZQ7 1/20 0.50
CYP3A4 P08684 1/20 0.50
THRB P10828 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25812119 0.88 LMNA (0.54) LMNAALDH1A1SLC22A2SLC22A1TSHR
SCHEMBL14537512 0.81 HDAC3 (0.56) ALDH1A1CYP2C19HDAC3HDAC1CD274
SCHEMBL30547775 0.77 MAOB (0.59) HDAC3HDAC1CD274MAOBCHRNA7
SCHEMBL1995821 0.77 MAOB (0.59) HDAC3HDAC1CD274MAOBCHRNA7
SCHEMBL15219324 0.76 ALDH1A1 (0.59) LMNAALDH1A1SLC22A2SLC22A1TSHR
SCHEMBL25811248 0.76 MAPT (0.62) LMNAALDH1A1SLC22A2SLC22A1TSHR
SCHEMBL13426153 0.75 LMNA (0.58) LMNAALDH1A1SLC22A2SLC22A1TSHR
SCHEMBL2442620 0.75 LMNA (0.58) LMNAALDH1A1SLC22A2SLC22A1TSHR
SCHEMBL11919098 0.75 LMNA (0.58) LMNAALDH1A1SLC22A2SLC22A1TSHR
SCHEMBL22043064 0.75 ALDH1A1 (0.74) LMNAALDH1A1SLC22A2SLC22A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1565455-A1 INDOLYL PYRAZINONE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS Bayer Pharmaceuticals Corporation (US) 2005-08-24 EP disclosed
WO-2004043950-A1 INDOLYL PYRAZINONE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER PHARMACEUTICALS CORPORATION (US) 2004-05-27 WO disclosed