SCHEMBL625201

SCHEMBL625201

NCC1CCCN(c2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)C1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.48
KCNH2 Q12809 5/20 0.41
MAP3K12 Q12852 3/20 0.39
PTPN11 Q06124 1/20 0.38
HASPIN Q8TF76 2/20 0.37
FLT3 P36888 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626391 0.92 PIK3CA (0.48) PIK3CAKCNH2MAP3K12
SCHEMBL624411 0.89 PIK3CA (0.54) PIK3CAKCNH2HASPINFLT3
SCHEMBL625018 0.88 PIK3CA (0.51) PIK3CAKCNH2HASPIN
SCHEMBL625432 0.86 PIK3CA (0.50) PIK3CAKCNH2MAP3K12HASPIN
SCHEMBL625202 0.86 MAP3K12 (0.43) MAP3K12
SCHEMBL625222 0.85 PIK3CA (0.48) PIK3CAKCNH2
SCHEMBL625227 0.84 PIK3CA (0.55) PIK3CAKCNH2MAP3K12HASPINFLT3
SCHEMBL625177 0.82 PIK3CA (0.49) PIK3CAKCNH2
SCHEMBL624865 0.82 PIK3CA (0.49) PIK3CAKCNH2
SCHEMBL627410 0.82 PIK3CA (0.57) PIK3CAKCNH2HASPINFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed