SCHEMBL624865

SCHEMBL624865

CC(=O)NC1CCCN(c2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)C1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 11/20 0.49
RIPK1 Q13546 1/20 0.43
KCNH2 Q12809 4/20 0.41
EIF2AK4 Q9P2K8 1/20 0.41
SYK P43405 1/20 0.41
BTK Q06187 1/20 0.40
PIK3CD O00329 2/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626006 0.90 PIK3CA (0.46) PIK3CARIPK1KCNH2PIK3CDPIK3CB
SCHEMBL624869 0.88 PIK3CA (0.52) PIK3CARIPK1KCNH2BTKPIK3CD
SCHEMBL624866 0.87 PIK3CA (0.46) PIK3CASYK
SCHEMBL625177 0.85 PIK3CA (0.49) PIK3CAKCNH2PIK3CD
SCHEMBL624990 0.85 PIK3CA (0.47) PIK3CARIPK1KCNH2SYK
SCHEMBL625222 0.84 PIK3CA (0.48) PIK3CAKCNH2PIK3CDPIK3CBPIK3CG
SCHEMBL625018 0.84 PIK3CA (0.51) PIK3CAKCNH2PIK3CDPIK3CBPIK3CG
SCHEMBL626391 0.83 PIK3CA (0.48) PIK3CAKCNH2
SCHEMBL625732 0.82 PIK3CA (0.53) PIK3CAKCNH2PIK3CDPIK3CBPIK3CG
SCHEMBL625201 0.82 PIK3CA (0.48) PIK3CAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed