SCHEMBL625177

SCHEMBL625177

CNC(=O)C1CCCN(c2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)C1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.49
PIK3CD O00329 3/20 0.44
KCNH2 Q12809 4/20 0.41
MAPT P10636 2/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625222 0.90 PIK3CA (0.48) PIK3CAPIK3CDKCNH2
SCHEMBL625178 0.87 MAPT (0.54) MAPTTHRB
SCHEMBL624633 0.86 PIK3CA (0.47) PIK3CAKCNH2MAPT
SCHEMBL624865 0.85 PIK3CA (0.49) PIK3CAPIK3CDKCNH2
SCHEMBL625018 0.84 PIK3CA (0.51) PIK3CAPIK3CDKCNH2
SCHEMBL626391 0.83 PIK3CA (0.48) PIK3CAKCNH2
SCHEMBL624869 0.83 PIK3CA (0.52) PIK3CAPIK3CDKCNH2
SCHEMBL625201 0.82 PIK3CA (0.48) PIK3CAKCNH2
SCHEMBL626006 0.82 PIK3CA (0.46) PIK3CAPIK3CDKCNH2MAPTTHRB
SCHEMBL625746 0.81 PIK3CA (0.54) PIK3CAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed