SCHEMBL625281

SCHEMBL625281

CN(c1nn2c(-c3cnc(N)c(C(F)(F)F)c3)cnc2s1)C1CCC(C)(O)CC1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.52
MAP3K12 Q12852 10/20 0.40
PIM1 P11309 1/20 0.37
KCNH2 Q12809 1/20 0.37
DLK1 P80370 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626636 0.90 PIK3CA (0.54) PIK3CAMAP3K12
SCHEMBL626638 0.90 PIK3CA (0.54) PIK3CAMAP3K12
SCHEMBL627785 0.86 PIK3CA (0.56) PIK3CAMAP3K12PIM1
SCHEMBL627784 0.86 PIK3CA (0.56) PIK3CAMAP3K12PIM1
SCHEMBL625653 0.86 PIK3CA (0.54) PIK3CAMAP3K12
SCHEMBL625050 0.85 PIK3CA (0.53) PIK3CAMAP3K12
SCHEMBL625863 0.84 PIK3CA (0.51) PIK3CAMAP3K12
SCHEMBL625282 0.84 MAP3K12 (0.45) PIK3CAMAP3K12DLK1
SCHEMBL625635 0.83 PIK3CA (0.51) PIK3CAPIM1KCNH2
SCHEMBL624921 0.81 PIK3CA (0.49) PIK3CAMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed