SCHEMBL625863

SCHEMBL625863

CN(c1nn2c(-c3cnc(N)c(C(F)(F)F)c3)cnc2s1)C1CCC(=NO)CC1

nearest known ligand 0.51

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 11/20 0.51
MAP3K12 Q12852 9/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625050 0.88 PIK3CA (0.53) PIK3CAMAP3K12
SCHEMBL626636 0.87 PIK3CA (0.54) PIK3CAMAP3K12
SCHEMBL626638 0.87 PIK3CA (0.54) PIK3CAMAP3K12
SCHEMBL625653 0.85 PIK3CA (0.54) PIK3CAMAP3K12
SCHEMBL625281 0.84 PIK3CA (0.52) PIK3CAMAP3K12
SCHEMBL625864 0.84 MAP3K12 (0.44) PIK3CAMAP3K12
SCHEMBL627785 0.83 PIK3CA (0.56) PIK3CAMAP3K12
SCHEMBL627784 0.83 PIK3CA (0.56) PIK3CAMAP3K12
SCHEMBL624921 0.80 PIK3CA (0.49) PIK3CAMAP3K12
SCHEMBL625862 0.80 PIK3CA (0.47) PIK3CAMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed