SCHEMBL625282

SCHEMBL625282

CN(c1nn2cc(-c3cnc(N)c(C(F)(F)F)c3)nc2s1)C1CCC(C)(O)CC1

nearest known ligand 0.45

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 19/20 0.45
PIK3CA P42336 1/20 0.43
DLK1 P80370 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626637 0.90 MAP3K12 (0.47) MAP3K12PIK3CADLK1
SCHEMBL627783 0.86 MAP3K12 (0.46) MAP3K12PIK3CADLK1
SCHEMBL625654 0.86 MAP3K12 (0.47) MAP3K12PIK3CADLK1
SCHEMBL625051 0.85 MAP3K12 (0.46) MAP3K12PIK3CADLK1
SCHEMBL625864 0.85 MAP3K12 (0.44) MAP3K12PIK3CADLK1
SCHEMBL625281 0.84 PIK3CA (0.52) MAP3K12PIK3CADLK1
SCHEMBL625636 0.83 MAP3K12 (0.44) MAP3K12PIK3CADLK1
SCHEMBL624922 0.81 PIK3CA (0.42) MAP3K12PIK3CA
SCHEMBL626135 0.81 PIK3CA (0.45) MAP3K12PIK3CADLK1
SCHEMBL625010 0.73 HSD11B1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed