SCHEMBL625291

SCHEMBL625291

FC(F)(F)Oc1cccc(-c2cnc3sc(NC4CCOCC4)nn23)c1

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 13/20 0.68
DYRK1A Q13627 2/20 0.58
FYN P06241 5/20 0.58
KCNH2 Q12809 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1945309 0.90 FYN (0.71) PIM1FYNKCNH2
Hydrochloric Acid SCHEMBL625022 0.89 FYN (0.58) PIM1FYNKCNH2
SCHEMBL626258 0.89 PIM1 (0.68) PIM1FYNKCNH2
SCHEMBL1944058 0.89 FYN (0.72) PIM1FYNKCNH2
SCHEMBL623434 0.88 FYN (0.57) PIM1FYNKCNH2
SCHEMBL1944167 0.86 PIM1 (0.70) PIM1DYRK1AFYNKCNH2
SCHEMBL625500 0.83 FYN (0.55) PIM1FYNKCNH2
SCHEMBL623872 0.82 FYN (0.52) PIM1FYNKCNH2
SCHEMBL625560 0.82 FYN (0.50) PIM1FYNKCNH2
SCHEMBL102533 0.81 PIM1 (1.00) PIM1DYRK1AFYNKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed