SCHEMBL6253124

SCHEMBL6253124

Cc1ccc(O)c(Cc2cc(C)cc(Cc3cc(C)ccc3O)c2C[C@H](N)C(=O)O)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 1/20 0.54
SLC7A5 Q01650 4/20 0.52
USP2 O75604 3/20 0.47
KDM4E B2RXH2 2/20 0.47
ALOX15 P16050 2/20 0.47
RECQL P46063 2/20 0.47
HIF1A Q16665 2/20 0.47
HSD17B10 Q99714 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
EGFR P00533 1/20 0.47
LCK P06239 1/20 0.47
FYN P06241 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
PTGS1 P23219 1/20 0.47
HTR2A P28223 1/20 0.47
PTGS2 P35354 1/20 0.47
THRB P10828 7/20 0.45
THRA P10827 5/20 0.45
LMNA P02545 3/20 0.45
MEN1 O00255 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2032864 0.85 THRB (0.62) AMY1ASLC7A5USP2KDM4EALOX15
SCHEMBL2033124 0.85 THRB (0.62) AMY1ASLC7A5USP2KDM4EALOX15
SCHEMBL2033125 0.85 THRB (0.62) AMY1ASLC7A5USP2KDM4EALOX15
SCHEMBL2028640 0.76 KDM4E (0.62) SLC7A5USP2KDM4EALOX15RECQL
SCHEMBL2028058 0.76 KDM4E (0.62) SLC7A5USP2KDM4EALOX15RECQL
SCHEMBL2028643 0.76 KDM4E (0.62) SLC7A5USP2KDM4EALOX15RECQL
SCHEMBL29621432 0.74 AMY1A (0.83) AMY1AUSP2ALOX15HIF1AHSD17B10
SCHEMBL29402131 0.74 AMY1A (0.83) AMY1AUSP2ALOX15HIF1AHSD17B10
SCHEMBL50622 0.74 AMY1A (0.83) AMY1AUSP2ALOX15HIF1AHSD17B10
SCHEMBL5288482 0.74 USP2 (0.50) SLC7A5USP2KDM4EALOX15RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1570002-A1 FLAME-RESISTANT POLYCARBONATE COMPOSITIONS COMPRISING PHOSPHORUS-SILICON COMPOUNDS Bayer MaterialScience AG (DE) 2005-09-07 EP disclosed
WO-2004052990-A1 FLAME-RESISTANT POLYCARBONATE COMPOSITIONS COMPRISING PHOSPHORUS-SILICON COMPOUNDS BAYER MATERIALSCIENCE AG (DE) 2004-06-24 WO disclosed
EP-1404750-A1 FLAME-PROOFED POLYESTER MOULDING MATERIALS WITH ZNS BAYER AG (DE) 2004-04-07 EP disclosed
EP-1355988-A1 POLYCARBONATE COMPOSITIONS HAVING A REDUCED IRON CONTENT Bayer Aktiengesellschaft (DE) 2003-10-29 EP disclosed
WO-2003002643-A1 FLAME-PROOFED POLYESTER MOULDING MATERIALS WITH ZNS BAYER AKTIENGESELLSCHAFT (DE) 2003-01-09 WO disclosed
EP-1230302-A2 POLYMER BLENDS CONTAINING MODIFIED POLYESTERS Bayer Aktiengesellschaft (DE) 2002-08-14 EP disclosed
WO-2002059203-A1 POLYCARBONATE COMPOSITIONS HAVING A REDUCED IRON CONTENT BAYER AKTIENGESELLSCHAFT (DE) 2002-08-01 WO disclosed
EP-1144511-A2 FLAME-RESISTANT POLYCARBONATE ABS MOULDING MATERIAL Bayer Aktiengesellschaft (DE) 2001-10-17 EP disclosed
WO-2001023474-A2 POLYMER BLENDS CONTAINING MODIFIED POLYESTERS BAYER AKTIENGESELLSCHAFT (DE) 2001-04-05 WO disclosed
WO-2000031173-A2 FLAME-RESISTANT POLYCARBONATE ABS MOULDING MATERIAL BAYER AKTIENGESELLSCHAFT (DE) 2000-06-02 WO disclosed