SCHEMBL625433

SCHEMBL625433

CS(=O)(=O)NCC1CCCN(c2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)C1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPT P10636 16/20 0.43
POLB P06746 1/20 0.43
THRB P10828 2/20 0.42
LMNA P02545 4/20 0.42
MAP3K12 Q12852 4/20 0.40
TP53 P04637 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626169 0.91 MAP3K12 (0.41) MAPTTHRBLMNAMAP3K12
SCHEMBL625432 0.88 PIK3CA (0.50) MAP3K12
SCHEMBL624870 0.87 MAPT (0.42) MAPTPOLBTHRBLMNAMAP3K12
SCHEMBL625202 0.86 MAP3K12 (0.43) MAPTPOLBTHRBLMNAMAP3K12
SCHEMBL626392 0.86 MAP3K12 (0.44) MAPTPOLBTHRBLMNAMAP3K12
SCHEMBL625733 0.83 MAP3K12 (0.42) MAPTPOLBTHRBMAP3K12
SCHEMBL625019 0.82 MAP3K12 (0.45) MAPTPOLBTHRBLMNAMAP3K12
SCHEMBL624968 0.82 MAP3K12 (0.43) MAPTTHRBMAP3K12
SCHEMBL625178 0.81 MAPT (0.54) MAPTPOLBTHRBLMNATP53
SCHEMBL624866 0.81 PIK3CA (0.46) MAPTPOLBTHRBLMNAMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed