SCHEMBL624968

SCHEMBL624968

CS(=O)(=O)NC1CCN(c2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 7/20 0.43
MAPT P10636 6/20 0.42
PIK3CA P42336 4/20 0.42
THRB P10828 3/20 0.40
GAA P10253 1/20 0.39
SMO Q99835 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625733 0.95 MAP3K12 (0.42) MAP3K12MAPTPIK3CATHRB
SCHEMBL624870 0.90 MAPT (0.42) MAP3K12MAPTPIK3CATHRB
SCHEMBL626169 0.88 MAP3K12 (0.41) MAP3K12MAPTPIK3CATHRBGAA
SCHEMBL624967 0.86 PIK3CA (0.55) MAP3K12PIK3CASMO
SCHEMBL627411 0.85 MAP3K12 (0.47) MAP3K12MAPTPIK3CA
SCHEMBL625621 0.84 MAP3K12 (0.46) MAP3K12MAPTPIK3CA
SCHEMBL626106 0.84 THRB (0.49) MAPTPIK3CATHRBGAA
SCHEMBL625132 0.84 CKS1B (0.42) MAP3K12MAPTPIK3CATHRBGAA
SCHEMBL627373 0.83 MAP3K12 (0.46) MAP3K12MAPTPIK3CATHRB
SCHEMBL626464 0.83 MAPT (0.47) MAP3K12MAPTPIK3CATHRBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed