SCHEMBL625733

SCHEMBL625733

CS(=O)(=O)NC1CCN(c2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)C1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 10/20 0.42
PIK3CA P42336 4/20 0.41
MAPT P10636 4/20 0.39
THRB P10828 2/20 0.38
IRAK1 P51617 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624870 0.95 MAPT (0.42) MAP3K12PIK3CAMAPTTHRBPOLB
SCHEMBL624968 0.95 MAP3K12 (0.43) MAP3K12PIK3CAMAPTTHRB
SCHEMBL625732 0.87 PIK3CA (0.53) MAP3K12PIK3CA
SCHEMBL626169 0.85 MAP3K12 (0.41) MAP3K12PIK3CAMAPTTHRB
SCHEMBL624991 0.84 SYK (0.45) MAP3K12PIK3CA
SCHEMBL625433 0.83 MAPT (0.43) MAP3K12MAPTTHRBPOLB
SCHEMBL625228 0.83 MAP3K12 (0.46) MAP3K12PIK3CA
SCHEMBL624866 0.83 PIK3CA (0.46) MAP3K12PIK3CAMAPTTHRBPOLB
SCHEMBL626620 0.82 MAP3K12 (0.52) MAP3K12PIK3CA
SCHEMBL624869 0.82 PIK3CA (0.52) MAP3K12PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed