SCHEMBL6254331

SCHEMBL6254331

CNC(=O)C#Cc1ccc(F)cc1.O=C(O)N1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.43
GPR183 P32249 9/20 0.42
ALOX5 P09917 1/20 0.40
TDP1 Q9NUW8 1/20 0.38
APP P05067 1/20 0.37
CHRM1 P11229 1/20 0.37
MCHR1 Q99705 1/20 0.37
GFER P55789 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6250333 0.99 GPR183 (0.43) KMT2AGPR183ALOX5APPGFER
SCHEMBL6258306 0.85 DPP4 (0.45) GPR183GFERALDH1A1
SCHEMBL666992 0.83 APP (0.49) KMT2AGPR183APPGFERALDH1A1
SCHEMBL6228346 0.77 KMT2A (0.43) KMT2AGPR183ALOX5TDP1ALDH1A1
SCHEMBL14737095 0.73 GRM3 (0.44) KMT2AGPR183ALDH1A1
Fluorobenzene SCHEMBL28159220 0.71 HPGD (0.55) KMT2AALOX5ALDH1A1
SCHEMBL16151536 0.70 HPGD (0.65) KMT2AGPR183ALDH1A1
SCHEMBL4554708 0.69 NPSR1 (0.55) KMT2AAPPGFERALDH1A1
SCHEMBL22031721 0.69 GRM5 (0.46) KMT2ATDP1ALDH1A1
SCHEMBL1840511 0.68 FABP4 (0.46) GPR183GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517894-A1 N-BENZYL-3-PHENYL-3-HETEROCYCLYL-PROPIONAMIDE COMPOUNDS AS TACHYKININ ANTAGONISTS AND/OR SEROTONIN REUPTAKE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-03-30 EP disclosed
WO-2004005255-A1 N-BENZYL-3-PHENYL-3-HETEROCYCLYL-PROPIONAMIDE COMPOUNDS AS TACHYKININ AND/ OR SEROTONIN REUPTAKE INHIBITORS GLAXO GROUP LIMITED (GB) 2004-01-15 WO disclosed