SCHEMBL6255368

SCHEMBL6255368

CC(C)(C)CN(Cc1cccc(-c2ccc(C=O)cc2)c1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGES O14684 2/20 0.48
BCHE P06276 1/20 0.44
AOC3 Q16853 11/20 0.43
BCL2 P10415 1/20 0.43
TRIM24 O15164 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
HSD17B1 P14061 1/20 0.40
HSD17B2 P37059 1/20 0.40
PTGS2 P35354 1/20 0.40
DRD1 P21728 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6184553 0.87 PTGES (0.52) PTGESBCHEAOC3BCL2TRIM24
SCHEMBL6032493 0.86 PTGES (0.51) PTGESAOC3BCL2HSD17B1HSD17B2
SCHEMBL2177213 0.82 MEN1 (0.47) PTGESBCHEAOC3BCL2TRIM24
SCHEMBL3948563 0.81 AOC3 (0.57) BCHEAOC3TRIM24TRIM33HSD17B1
SCHEMBL6185834 0.79 AOC3 (0.58) PTGESBCHEAOC3BCL2TRIM24
SCHEMBL6472820 0.79 AOC3 (0.49) PTGESBCHEAOC3HSD17B2DRD1
SCHEMBL6182236 0.77 HSD17B2 (0.62) BCHEAOC3HSD17B1HSD17B2
SCHEMBL6184104 0.76 BCHE (0.53) PTGESBCHEAOC3BCL2HSD17B1
SCHEMBL7025759 0.76 GRIN2D (0.43) PTGES
SCHEMBL7021355 0.76 PTGES (0.43) PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567509-A2 BIPHENYL COMPOUNDS WHICH ACTIVATE PPAR-GAMMA TYPE RECEPTORS, AND USE THEREOF IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS Galderma Research & Development, S.N.C. (FR) 2005-08-31 EP disclosed
US-6927228-B2 Biphenyl compounds usefuf in treatment of human and veterinary medicines such as dermatology, cardivovascular diseases, immune diseases or diseases associated with lipid metabolisms, or in cosmetic formulation GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2005-08-09 US disclosed
WO-2004048351-A2 BIPHENYL COMPOUNDS WHICH ACTIVATE PPAR-GAMMA TYPE RECEPTORS AND USE THEREOF IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2004-06-10 WO disclosed
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors GALDERMA RESEARCH & DEVELOPMENT S.N.C. (FR) 2004-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors PPARG, PPARA, PPARD PTGES 520/4885BCHE 1768/4885AOC3 1747/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.