SCHEMBL625753

SCHEMBL625753

CC(C)S(=O)(=O)N1CCC(Nc2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)CC1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.49
FYN P06241 9/20 0.44
HASPIN Q8TF76 1/20 0.42
MAP3K12 Q12852 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626206 0.91 PIK3CA (0.53) PIK3CAFYNHASPINMAP3K12
SCHEMBL624427 0.84 PIK3CA (0.50) PIK3CAFYNHASPINMAP3K12
SCHEMBL625300 0.82 PIK3CA (0.51) PIK3CAFYNHASPIN
SCHEMBL627398 0.82 PIK3CA (0.53) PIK3CAFYNHASPIN
SCHEMBL627396 0.82 PIK3CA (0.53) PIK3CAFYNHASPIN
SCHEMBL625455 0.82 PIK3CA (0.43) PIK3CAFYNHASPINMAP3K12
SCHEMBL627441 0.81 FYN (0.63) PIK3CAFYNHASPIN
SCHEMBL625235 0.81 FYN (0.52) PIK3CAFYNHASPIN
SCHEMBL627439 0.81 FYN (0.63) PIK3CAFYNHASPIN
SCHEMBL625127 0.81 PIK3CA (0.48) PIK3CAFYNHASPIN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed