SCHEMBL625862

SCHEMBL625862

Nc1ncc(-c2cnc3sc(CNC4CCC(=NO)CC4)nn23)cc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.47
MAP3K12 Q12852 8/20 0.36
PIM1 P11309 1/20 0.35
PIK3CD O00329 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625652 0.86 PIK3CA (0.49) PIK3CAMAP3K12PIK3CDPIK3CBFYN
SCHEMBL625280 0.84 PIK3CA (0.49) PIK3CAMAP3K12PIM1
SCHEMBL626133 0.81 PIK3CA (0.47) PIK3CAMAP3K12PIK3CDPIK3CBPIK3CG
SCHEMBL624920 0.80 PIK3CA (0.46) PIK3CAPIK3CD
SCHEMBL625863 0.80 PIK3CA (0.51) PIK3CAMAP3K12
SCHEMBL625300 0.73 PIK3CA (0.51) PIK3CAFYN
SCHEMBL627439 0.72 FYN (0.63) PIK3CAFYN
SCHEMBL627441 0.72 FYN (0.63) PIK3CAFYN
SCHEMBL627610 0.71 FYN (0.56) PIK3CAFYN
SCHEMBL627612 0.71 FYN (0.56) PIK3CAFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed