SCHEMBL6259634

SCHEMBL6259634

NC(=O)c1ccc(-c2nc3ccc(F)cc3[nH]2)cc1

nearest known ligand 0.82

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 18/20 0.82
NR4A2 P43354 1/20 0.69
PKN1 Q16512 1/20 0.65
PKN2 Q16513 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6247109 0.89 CHEK2 (0.70) CHEK2NR4A2PKN1PKN2
SCHEMBL20982670 0.87 CHEK2 (0.86) CHEK2PKN1PKN2
SCHEMBL27528263 0.84 MEN1 (0.74) CHEK2PKN1PKN2
Terephthalamide SCHEMBL28143925 0.83 CHEK2 (0.75) CHEK2PKN1PKN2
SCHEMBL6260767 0.83 MMP2 (0.78) CHEK2PKN1PKN2
SCHEMBL3922046 0.82 CHEK2 (0.81) CHEK2NR4A2PKN1PKN2
SCHEMBL30938560 0.82 NR4A2 (1.00) CHEK2NR4A2
SCHEMBL24312910 0.81 PLAU (0.71) CHEK2PKN1PKN2
SCHEMBL29557707 0.81 PLAU (0.71) CHEK2PKN1PKN2
SCHEMBL6259639 0.81 SMN1; SMN2 (0.76) CHEK2NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005030206-A1 ARYL-1,3-AZOLE DERIVATIVES AND METHODS FOR INHIBITING HEPARNASE ACTIVITY IMCLONE SYSTEMS INCORPORATED (US) 2005-04-07 WO disclosed