SCHEMBL6259696

SCHEMBL6259696

NC(=O)n1c(-c2ccccc2)nc2c[c]ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
HSD17B10 Q99714 1/20 0.40
JAK2 O60674 2/20 0.38
JAK1 P23458 2/20 0.38
TYK2 P29597 2/20 0.38
JAK3 P52333 2/20 0.38
CNR2 P34972 1/20 0.37
KMT2A Q03164 3/20 0.36
PARP1 P09874 1/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
HTT P42858 1/20 0.36
ALDH1A1 P00352 2/20 0.35
PDE6D O43924 1/20 0.35
ALDH2 P05091 1/20 0.35
ALDH3A1 P30838 1/20 0.35
MAOA P21397 1/20 0.35
RAB9A P51151 4/20 0.35
NPC1 O15118 2/20 0.35
MEN1 O00255 2/20 0.35
CYP1A2 P05177 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6890976 0.82 KDM4E (0.56) KDM4EHSD17B10JAK2JAK1TYK2
SCHEMBL7945632 0.77 CNR2 (0.39) KDM4ECNR2HTTALDH1A1RAB9A
SCHEMBL2364958 0.75 PDE2A (0.38) KDM4EJAK2JAK1TYK2JAK3
SCHEMBL7048551 0.75 KDM4E (0.37) KDM4EHSD17B10KMT2ASMN1; SMN2HTT
SCHEMBL731625 0.75 ATM (0.56) KDM4EHSD17B10KMT2ASMN1; SMN2HTT
SCHEMBL732846 0.74 ESR1 (0.54) KMT2AHTTALDH1A1PDE6DALDH2
SCHEMBL2338761 0.73 CYP2C9 (0.34) KMT2AHTTMEN1CYP1A2CYP2C19
SCHEMBL29145105 0.72 KDM4E (0.56) KDM4EHSD17B10JAK2JAK1TYK2
SCHEMBL28646061 0.72 ESR1 (0.52) KDM4EHSD17B10JAK2JAK1TYK2
SCHEMBL2105982 0.72 HSD17B10 (0.40) KDM4EHSD17B10CNR2SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005030206-A1 ARYL-1,3-AZOLE DERIVATIVES AND METHODS FOR INHIBITING HEPARNASE ACTIVITY IMCLONE SYSTEMS INCORPORATED (US) 2005-04-07 WO disclosed