SCHEMBL6260764

SCHEMBL6260764

C[C@H](N)C(=O)Nc1ccc(-c2c3ccccc3nc3ccccc23)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.67
ALDH1A1 P00352 3/20 0.53
GAA P10253 1/20 0.53
LTA4H P09960 1/20 0.49
IDO1 P14902 2/20 0.48
CIT O14578 1/20 0.47
KDM4E B2RXH2 4/20 0.47
KMT2A Q03164 3/20 0.47
POLB P06746 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
KDM1A O60341 1/20 0.47
MITF O75030 1/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
RAD52 P43351 1/20 0.47
RECQL P46063 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
XIAP P98170 4/20 0.45
NPC1 O15118 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5273543 0.84 CIT (0.50) TAAR1ALDH1A1GAACITKDM4E
SCHEMBL29226582 0.81 KMT2A (0.68) TAAR1ALDH1A1KDM4EKMT2APOLB
SCHEMBL1246982 0.81 TAAR1 (0.59) TAAR1ALDH1A1GAALTA4HCIT
SCHEMBL4652086 0.81 TAAR1 (1.00) TAAR1ALDH1A1LTA4HIDO1CIT
SCHEMBL1751436 0.81 TAAR1 (1.00) TAAR1ALDH1A1LTA4HIDO1CIT
SCHEMBL5273957 0.80 ACHE (0.63) TAAR1LTA4HIDO1CITXIAP
SCHEMBL5278210 0.80 TAAR1 (0.53) TAAR1ALDH1A1GAALTA4HIDO1
Hydrochloric Acid SCHEMBL5404008 0.79 ACHE (0.62) TAAR1LTA4HIDO1CITXIAP
Hydrochloric Acid SCHEMBL5414835 0.78 ACHE (0.60) TAAR1LTA4HIDO1CITXIAP
SCHEMBL5273024 0.78 JAK2 (0.50) ALDH1A1GAAKDM4EKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1587793-A1 ENZYME SUBSTRATES, CULTURE MEDIA CONTAINING SAME AND USE THEREOF IN ORDER TO DETECT AMINOPEPTIDASE ACTIVITY AND/OR DIFFERENTIATE GRAM-POSITIVE BACTERIA FROM GRAM-NEGATIVE BACTERIA BIOMERIEUX (FR) 2005-10-26 EP disclosed
WO-2004069804-A1 ENZYME SUBSTRATES, CULTURE MEDIA CONTAINING SAME AND USE THEREOF IN ORDER TO DETECT AMINOPEPTIDASE ACTIVITY AND/OR DIFFERENTIATE GRAM-POSITIVE BACTERIA FROM GRAM-NEGATIVE BACTERIA BIOMERIEUX (FR) 2004-08-19 WO disclosed