SCHEMBL6262602

SCHEMBL6262602

NS(=O)(=O)c1ccc(-c2cnn(-c3ccc(Cl)cc3)c2-c2ccccc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.71
PTGS1 P23219 12/20 0.71
LMNA P02545 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
CA1 P00915 2/20 0.55
CA2 P00918 2/20 0.55
CA4 P22748 2/20 0.55
CA9 Q16790 2/20 0.55
KDM4E B2RXH2 1/20 0.54
GAA P10253 1/20 0.54
HTT P42858 1/20 0.54
MEN1 O00255 1/20 0.53
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765046 0.96 PTGS2 (0.67) PTGS2PTGS1LMNANPSR1CA1
SCHEMBL8765473 0.95 PTGS2 (0.76) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765227 0.85 PTGS2 (0.62) PTGS2PTGS1LMNANPSR1KDM4E
SCHEMBL8633382 0.84 PTGS2 (0.65) PTGS2PTGS1LMNANPSR1CA1
SCHEMBL8765541 0.84 PTGS2 (0.62) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765203 0.83 PTGS2 (0.65) PTGS2PTGS1LMNANPSR1KDM4E
SCHEMBL3245704 0.83 PTGS2 (0.80) PTGS2PTGS1CA1CA2CA4
SCHEMBL213767 0.83 PTGS2 (1.00) PTGS2PTGS1CA1CA2CA4
SCHEMBL8765024 0.83 RAB9A (0.69) PTGS2PTGS1LMNANPSR1KDM4E
SCHEMBL6405376 0.82 PTGS2 (1.00) PTGS2PTGS1CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005044194-A2 TREATMENT OR PREVENTION OF NEOPLASIA BY USE OF AN Hsp90 INHIBITOR PHARMACIA CORPORATION (US) 2005-05-19 WO disclosed