SCHEMBL626456

SCHEMBL626456

CCCCn1cc(C=O)nn1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 4/20 0.44
AMY1A P0DUB6 1/20 0.40
P2RX7 Q99572 1/20 0.40
EPHX2 P34913 1/20 0.38
GBA1 P04062 5/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28267000 0.93 SMPD1 (0.52) SMPD1EPHX2GBA1
SCHEMBL24569915 0.89 P2RX7 (0.42) SMPD1P2RX7GBA1
SCHEMBL19165673 0.81 P2RX7 (0.37) SMPD1P2RX7
SCHEMBL18707087 0.81
SCHEMBL3744192 0.78 EP300 (0.47)
SCHEMBL24345690 0.76 P2RX7 (0.38) P2RX7
SCHEMBL5490200 0.75 SMPD1 (0.44) SMPD1EPHX2GBA1
SCHEMBL23636794 0.75 HDAC3 (0.46)
SCHEMBL28260567 0.75 HDAC3 (0.41) SMPD1EPHX2
SCHEMBL11899559 0.74 P2RX7 (0.42) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109096211-B Preparation method of polysubstituted triazole derivative 华侨大学 2021-11-23 CN disclosed
CN-109096211-A A kind of preparation method of polysubstituted triazole derivatives 华侨大学 2018-12-28 CN disclosed
US-20170210698-A1 COMPOUNDS AND COMPOSITIONS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC AGENTS ARES CAPITAL CORPORATION, AS AGENT 2017-07-27 US disclosed
WO-2012021390-A1 LIGANDS AND METHODS FOR LABELING BIOMOLECULES IN VIVO ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2012-02-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170210698-A1 COMPOUNDS AND COMPOSITIONS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC AGENTS LNPK, PLTP, PLIN3 SMPD1 26/4885AMY1A 4766/4885P2RX7 4727/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.