SCHEMBL626462

SCHEMBL626462

Nc1ncc(-c2cn3nc(N4CCCC5(CCN(S(=O)(=O)c6ccc(F)cc6F)CC5)C4)sc3n2)cc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.40
MAPT P10636 8/20 0.36
TNF P01375 2/20 0.36
SPR P35270 1/20 0.36
PIK3CA P42336 2/20 0.36
F2RL3 Q96RI0 1/20 0.35
LMNA P02545 1/20 0.34
MAP3K12 Q12852 4/20 0.33
HASPIN Q8TF76 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626461 0.89 PIK3CA (0.47) PKMPIK3CAHASPIN
SCHEMBL625703 0.83 MAP3K12 (0.44) PIK3CAF2RL3MAP3K12
SCHEMBL626243 0.81 MAP3K12 (0.46) PIK3CAF2RL3MAP3K12
SCHEMBL626123 0.80 RET (0.43) PIK3CAMAP3K12
SCHEMBL625459 0.74 MAP3K12 (0.41) PIK3CAF2RL3MAP3K12
SCHEMBL627020 0.74 RET (0.40) PIK3CAF2RL3MAP3K12
SCHEMBL626263 0.73 TNF (0.42) MAPTTNFPIK3CAMAP3K12
SCHEMBL624439 0.73 MAP3K12 (0.41) PIK3CAMAP3K12
SCHEMBL627432 0.71 RET (0.40) PIK3CAMAP3K12
SCHEMBL625702 0.71 PIK3CA (0.50) PIK3CAMAP3K12HASPIN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed