SCHEMBL627432

SCHEMBL627432

CC(C)(C)OC(=O)N1CCC2(CC1)CCN(c1nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s1)CC2

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RET P07949 2/20 0.40
PIK3CA P42336 3/20 0.40
MAP3K12 Q12852 13/20 0.39
PIK3R1 P27986 1/20 0.38
CYP11B2 P19099 1/20 0.38
DLK1 P80370 1/20 0.37
MAP4K1 Q92918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627020 0.94 RET (0.40) RETPIK3CAMAP3K12PIK3R1
SCHEMBL625422 0.93 PIK3CA (0.42) RETPIK3CAMAP3K12
SCHEMBL626123 0.92 RET (0.43) RETPIK3CAMAP3K12PIK3R1
SCHEMBL627431 0.87 PIK3CA (0.48) PIK3CA
SCHEMBL625408 0.86 MAP4K1 (0.39) PIK3CAMAP3K12DLK1MAP4K1
SCHEMBL627309 0.85 MAP3K12 (0.46) PIK3CAMAP3K12DLK1MAP4K1
SCHEMBL624439 0.83 MAP3K12 (0.41) PIK3CAMAP3K12DLK1
SCHEMBL626246 0.83 MAP3K12 (0.40) PIK3CAMAP3K12DLK1
SCHEMBL627019 0.82 PIK3CA (0.47) RETPIK3CAMAP3K12
SCHEMBL625132 0.81 CKS1B (0.42) RETPIK3CAMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed