SCHEMBL6265407

SCHEMBL6265407

O=C(O)c1ccc(OCC2CC(=O)N(c3ccccc3)C2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.48
USP2 O75604 1/20 0.48
TSHR P16473 1/20 0.48
GLA P06280 1/20 0.47
PKM P14618 2/20 0.47
MAPT P10636 1/20 0.47
MAPK1 P28482 1/20 0.47
GRM2 Q14416 4/20 0.45
POLB P06746 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
NR4A1 P22736 1/20 0.43
NR4A2 P43354 1/20 0.43
NR4A3 Q92570 1/20 0.43
CTSG P08311 1/20 0.43
CMA1 P23946 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6272688 0.95 ALDH1A1 (0.48) TP53USP2TSHRGLAPOLB
SCHEMBL6267136 0.91 NR4A1 (0.56) TP53USP2TSHRGLAPOLB
SCHEMBL6266719 0.90 ALDH1A1 (0.45) TP53USP2TSHRGLAPOLB
SCHEMBL6271800 0.90 GLA (0.46) TP53USP2TSHRGLAPOLB
SCHEMBL6267362 0.89 LMNA (0.55) TP53USP2TSHRGLAGRM2
SCHEMBL1060992 0.89 NPC1 (0.53) TP53USP2TSHRMAPTPOLB
SCHEMBL9031178 0.89 ALDH1A1 (0.53) TP53USP2TSHRMAPTMAPK1
SCHEMBL6270830 0.89 MAPT (0.47) TP53USP2TSHRGLAMAPT
SCHEMBL6269203 0.89 ALDH1A1 (0.58) TP53USP2TSHRPKMMAPT
SCHEMBL6272305 0.89 KMT2A (0.53) TP53USP2TSHRMAPTGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000620-B1 Lp(a)-LOWERING AGENTS AND APOPROTEIN (a) PRODUCTION INHIBITORS TAIHO PHARMACEUTICAL CO LTD (JP) 2005-12-07 EP disclosed
US-6166036-A Lp(a)-lowering agent and apolipoprotein (a) formation suppressing agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2000-12-26 US disclosed
EP-1000620-A1 Lp(a)-LOWERING AGENTS AND APOPROTEIN (a) PRODUCTION INHIBTORS TAIHO PHARMACEUTICAL COMPANY, LIMITED (JP) 2000-05-17 EP disclosed
EP-0393607-B1 Phenylcarboxylic acid derivatives having a hetero ring OTSUKA PHARMA CO LTD (JP) 1996-02-21 EP disclosed
US-5145865-A Fatty acid, cholesterol synthesis inhibitors; enzyme inhibitors; antilipemic agents OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1992-09-08 US disclosed
EP-0393607-A2 Phenylcarboxylic acid derivatives having a hetero ring OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-10-24 EP disclosed