SCHEMBL6268087

SCHEMBL6268087

CC(C)C(=O)Cn1cnc2c(=O)[nH]c(N)nc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TK1 P04183 2/20 0.58
MEN1 O00255 2/20 0.58
BLM P54132 2/20 0.58
KMT2A Q03164 2/20 0.58
ALDH1A1 P00352 1/20 0.58
LMNA P02545 1/20 0.58
CYP3A4 P08684 1/20 0.58
NFKB1 P19838 1/20 0.58
VCP P55072 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
HIF1A Q16665 1/20 0.58
PNP P00491 6/20 0.57
HBB P68871 2/20 0.57
USP2 O75604 1/20 0.57
TSHR P16473 1/20 0.57
EDNRA P25101 1/20 0.57
HTR2A P28223 1/20 0.57
RECQL P46063 1/20 0.57
HSD17B10 Q99714 1/20 0.57
MAPK1 P28482 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6271393 0.87 TK1 (0.58) TK1MEN1BLMKMT2AALDH1A1
SCHEMBL6265339 0.85 TK1 (0.62) TK1MEN1BLMKMT2AALDH1A1
SCHEMBL10919931 0.85 BLM (0.62) TK1MEN1BLMKMT2AALDH1A1
SCHEMBL10918874 0.84 BLM (0.61) TK1MEN1BLMKMT2AALDH1A1
SCHEMBL455494 0.84 PNP (0.64) TK1MEN1BLMKMT2AALDH1A1
SCHEMBL27667781 0.83 TK1 (0.60) TK1MEN1BLMKMT2AALDH1A1
SCHEMBL9463576 0.83 BLM (0.72) TK1MEN1BLMKMT2AALDH1A1
SCHEMBL6265535 0.82 TK1 (0.61) TK1MEN1BLMKMT2AALDH1A1
SCHEMBL7262060 0.82 HPRT1 (0.61) TK1MEN1BLMKMT2AALDH1A1
SCHEMBL7268685 0.82 HPRT1 (0.61) TK1MEN1BLMKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1017394-B1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER REC TECH LTD (GB) 2005-12-07 EP disclosed
US-6303618-B1 ADMINISTERING PURINE COMPOUND WHICH INHIBITS CYCLIC DEPENDENT KINASE ACTIVITY FOR THERAPY OF TUMOR OR OTHER CELL PROLIFERATION DISORDER CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2001-10-16 US disclosed
WO-1999002162-A9 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RES CAMPAIGN TECH (GB) 1999-07-29 WO disclosed