SCHEMBL6269623

SCHEMBL6269623

O=C(CCc1cccnc1)NCCCCN1CCC(C(=O)Nc2cccc3ccccc23)CC1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.46
HSD17B10 Q99714 2/20 0.46
ALDH1A1 P00352 4/20 0.43
LMNA P02545 3/20 0.43
TP53 P04637 1/20 0.43
DRD4 P21917 2/20 0.43
USP2 O75604 1/20 0.43
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CCR2 P41597 1/20 0.42
PTAFR P25105 1/20 0.41
TSHR P16473 1/20 0.41
SIGMAR1 Q99720 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL83396 0.87 KDM4E (0.54) KDM4EHSD17B10ALDH1A1LMNAUSP2
SCHEMBL3458647 0.81 HTR2A (0.54) KDM4EALDH1A1CYP2C9CYP2C19CYP1A2
SCHEMBL3073525 0.80 NAMPT (0.47) KDM4EHSD17B10ALDH1A1LMNAUSP2
SCHEMBL7672874 0.77 CHRNA7 (0.57) ALDH1A1LMNACYP2C9CYP2C19CYP1A2
SCHEMBL6271049 0.75 OPRL1 (0.46) ALDH1A1LMNACYP2C9CYP2C19CYP1A2
SCHEMBL82729 0.75 ALDH1A1 (0.54) ALDH1A1LMNACYP2C9CYP2C19CYP1A2
SCHEMBL3458409 0.74 ALDH1A1 (0.63) KDM4EALDH1A1CYP2C9CYP2C19CYP1A2
SCHEMBL3458346 0.73 DRD2 (0.54) ALDH1A1PTAFR
SCHEMBL5557428 0.73 DRD2 (0.48) ALDH1A1LMNACYP2C9CYP2C19CYP1A2
SCHEMBL3077208 0.72 FNTA (0.47) ALDH1A1CYP2C9CYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1079832-B1 USE OF VITAMIN PP COMPOUNDS KLINGE CO CHEM PHARM FAB (DE) 2005-11-30 EP claimed