SCHEMBL6270434

SCHEMBL6270434

CN(C)CCC1=C(CCc2cnccn2)c2ccc(C#N)cc2C1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 18/20 0.63
CYP2D6 P10635 17/20 0.63
KCNH2 Q12809 11/20 0.63
CHRM1 P11229 5/20 0.58
HTR2A P28223 1/20 0.58
CYP3A4 P08684 1/20 0.48
CHRM2 P08172 2/20 0.45
CHRM4 P08173 2/20 0.45
CHRM5 P08912 2/20 0.45
CHRM3 P20309 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6265065 0.81 HRH1 (0.62) HRH1CYP2D6KCNH2CHRM1HTR2A
SCHEMBL6414581 0.80 HRH1 (0.74) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6272080 0.77 CYP2D6 (1.00) HRH1CYP2D6KCNH2CHRM1HTR2A
SCHEMBL6265258 0.76 HRH1 (0.73) HRH1CYP2D6KCNH2CHRM1HTR2A
SCHEMBL6278779 0.73 HRH1 (1.00) HRH1CYP2D6KCNH2CHRM1HTR2A
SCHEMBL6417406 0.70 HRH1 (0.75) HRH1CYP2D6KCNH2CHRM1CHRM2
SCHEMBL2491068 0.68 HRH1 (0.50) HRH1CYP2D6KCNH2CHRM1HTR2A
SCHEMBL6416790 0.64 HRH1 (1.00) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL6276773 0.64 HRH1 (1.00) HRH1CYP2D6KCNH2CHRM1HTR2A
SCHEMBL3964757 0.62 HRH1 (0.45) HRH1CYP2D6KCNH2CHRM1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005097093-A1 SLEEP INDUCING COMPOUNDS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES, INC. (US) 2005-10-20 WO disclosed