SCHEMBL627086

SCHEMBL627086

OC(c1ncccn1)C1(c2cccc(OCC(F)(F)F)c2)CCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.49
GRIN2A Q12879 1/20 0.49
GRIN2B Q13224 1/20 0.49
TRPV3 Q8NET8 2/20 0.40
GPR3 P46089 1/20 0.36
CYP17A1 P05093 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CTSA P10619 1/20 0.35
CETP P11597 1/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
SIGMAR1 Q99720 1/20 0.33
EPHX2 P34913 1/20 0.33
NR1I2 O75469 1/20 0.33
ALDH1A1 P00352 1/20 0.32
RAB9A P51151 1/20 0.32
GRM2 Q14416 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624777 0.86 NR1I2 (0.43) GRIN1GRIN2AGRIN2BTRPV3CETP
SCHEMBL627085 0.84 TRPV3 (0.38) GRIN1GRIN2AGRIN2BTRPV3CETP
SCHEMBL624615 0.77 TRPV3 (0.46) TRPV3CYP2C9CYP2C19ALDH1A1HDAC6
SCHEMBL624513 0.75 TRPV3 (0.43) TRPV3NR1I2HDAC6
SCHEMBL624514 0.75 TRPV3 (0.43) TRPV3NR1I2HDAC6
SCHEMBL625376 0.75 TRPV3 (0.43) TRPV3NR1I2HDAC6
SCHEMBL624825 0.74 NR1I2 (0.57) TRPV3NR1I2
SCHEMBL624452 0.74 NR1I2 (0.59) TRPV3CETPNR1I2HDAC6
SCHEMBL624746 0.72 TRPV3 (0.49) TRPV3CYP17A1NR1I2HDAC6
SCHEMBL14893409 0.71 NR1I2 (0.39) TRPV3CETPNR1I2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2603490-A1 NOVEL TRPV3 MODULATORS AbbVie Inc. (US) 2013-06-19 EP disclosed
WO-2012019315-A1 NOVEL TRPV3 MODULATORS ABBOTT LABORATORIES (US) 2012-02-16 WO disclosed