SCHEMBL6270933

SCHEMBL6270933

COC(=O)C1CC(=O)N(c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.60
CA2 P00918 3/20 0.60
CA4 P22748 3/20 0.60
CA6 P23280 3/20 0.60
CA7 P43166 3/20 0.60
CA9 Q16790 3/20 0.60
CA13 Q8N1Q1 3/20 0.60
ALDH1A1 P00352 3/20 0.60
CA5B Q9Y2D0 2/20 0.60
CA12 O43570 1/20 0.60
CA14 Q9ULX7 1/20 0.60
GAA P10253 1/20 0.60
SMN1; SMN2 Q16637 2/20 0.55
KMT2A Q03164 2/20 0.55
MEN1 O00255 1/20 0.55
LMNA P02545 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C19 P33261 1/20 0.55
MAPT P10636 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6265330 0.85 ALDH1A1 (0.70) CA1CA2CA4CA6CA7
SCHEMBL6272177 0.84 KMT2A (0.64) CA1CA2CA4CA6CA7
SCHEMBL7825178 0.83 TSHR (0.66) CA1CA2CA4CA6CA7
SCHEMBL6273571 0.83 ALDH1A1 (0.62) CA1CA2CA4CA6CA7
SCHEMBL19793283 0.81 MAPK1 (0.70) CA1CA2CA4CA6CA7
SCHEMBL1777398 0.81 ALDH1A1 (0.70) CA1CA2CA4CA6CA7
SCHEMBL9031939 0.81 MAPK1 (0.70) CA1CA2CA4CA6CA7
SCHEMBL3365627 0.81 ALDH1A1 (0.70) CA1CA2CA4CA6CA7
SCHEMBL3365457 0.81 ALDH1A1 (0.70) CA1CA2CA4CA6CA7
SCHEMBL3366104 0.81 CA1 (0.67) CA1CA2CA4CA6CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000620-B1 Lp(a)-LOWERING AGENTS AND APOPROTEIN (a) PRODUCTION INHIBITORS TAIHO PHARMACEUTICAL CO LTD (JP) 2005-12-07 EP disclosed
US-6166036-A Lp(a)-lowering agent and apolipoprotein (a) formation suppressing agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2000-12-26 US disclosed
EP-1000620-A1 Lp(a)-LOWERING AGENTS AND APOPROTEIN (a) PRODUCTION INHIBTORS TAIHO PHARMACEUTICAL COMPANY, LIMITED (JP) 2000-05-17 EP disclosed
EP-0393607-B1 Phenylcarboxylic acid derivatives having a hetero ring OTSUKA PHARMA CO LTD (JP) 1996-02-21 EP disclosed
US-5145865-A Fatty acid, cholesterol synthesis inhibitors; enzyme inhibitors; antilipemic agents OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1992-09-08 US disclosed
EP-0393607-A2 Phenylcarboxylic acid derivatives having a hetero ring OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-10-24 EP disclosed