SCHEMBL627167

SCHEMBL627167

CS(=O)(=O)N1CCC(Nc2nn3c(I)cnc3s2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 10/20 0.46
KCNH2 Q12809 1/20 0.42
CCNE1 P24864 5/20 0.41
CDK2 P24941 5/20 0.41
CCNB2 O95067 3/20 0.41
CCNE2 O96020 3/20 0.41
CDK1 P06493 3/20 0.41
CCNB1 P14635 3/20 0.41
CDK5 Q00535 3/20 0.41
CDK5R1 Q15078 3/20 0.41
CCNB3 Q8WWL7 3/20 0.41
HASPIN Q8TF76 1/20 0.40
JAK2 O60674 1/20 0.40
JAK3 P52333 1/20 0.40
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
CCNT1 O60563 1/20 0.39
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39
CDK9 P50750 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627199 0.84 FYN (0.46) FYNCDK2HASPINJAK2JAK3
SCHEMBL624132 0.83 MKNK1 (0.48) FYNKCNH2CCNE1CDK2CCNE2
SCHEMBL626175 0.79 FYN (0.46) FYNHASPIN
SCHEMBL627492 0.79 CDK2 (0.39) FYNKCNH2CCNE1CDK2CCNB2
SCHEMBL627493 0.79 CCNE1 (0.37) FYNKCNH2CCNE1CDK2CCNB2
SCHEMBL626171 0.79 FYN (0.54) FYNKCNH2HASPIN
SCHEMBL628243 0.78 FYN (0.46) FYNHASPIN
SCHEMBL627017 0.77 FYN (0.47) FYNHASPIN
SCHEMBL627018 0.77 FYN (0.47) FYNHASPIN
SCHEMBL627849 0.77 FYN (0.46) FYNKCNH2HASPINJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed