SCHEMBL6273585

SCHEMBL6273585

C[C@@H]1CN(c2nccc3[nH]ccc23)CCN1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.47
JAK3 P52333 4/20 0.43
LCK P06239 1/20 0.39
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
HTR2C P28335 4/20 0.39
HRH4 Q9H3N8 2/20 0.39
ACVR1 Q04771 1/20 0.39
ATR Q13535 1/20 0.38
ATRIP Q8WXE1 1/20 0.38
ROCK2 O75116 1/20 0.38
PRKCQ Q04759 1/20 0.38
PRKCD Q05655 1/20 0.38
DOT1L Q8TEK3 2/20 0.38
ADRB1 P08588 1/20 0.38
HTR6 P50406 1/20 0.38
JAK2 O60674 2/20 0.36
JAK1 P23458 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6638364 0.80 HTR2C (0.59) HTR2CHRH4ROCK2ADRB1HTR6
Hydrochloric Acid SCHEMBL6643702 0.79 HTR2C (0.57) HTR2CHRH4ROCK2ADRB1HTR6
SCHEMBL20157192 0.78 KIT (0.42) KITJAK3MAPK13MAPK12MAPK11
SCHEMBL20157193 0.78 KIT (0.42) KITJAK3MAPK13MAPK12MAPK11
SCHEMBL6271843 0.77 HTR2C (0.65) KITHTR2CHRH4PRKCQPRKCD
SCHEMBL6281370 0.77 HTR2C (0.65) KITHTR2CHRH4PRKCQPRKCD
SCHEMBL3690829 0.76 HTR2C (0.66) KITMAPK13MAPK12MAPK11MAPK14
SCHEMBL18437145 0.76 HRH4 (0.55) JAK3HRH4ROCK2HTR6
SCHEMBL30146614 0.75 ADRB1 (0.64) HTR2CADRB1HTR6
SCHEMBL3678498 0.75 HTR2C (0.67) KITHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005121094-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES AS ANTI-HIV-AGENTS PFIZER LIMITED (GB) 2005-12-22 WO disclosed