SCHEMBL627456

SCHEMBL627456

Nc1ncc(-c2cnc3sc(N[C@H]4CC[C@H](NS(=O)(=O)c5ccc(F)cc5F)CC4)nn23)cc1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FYN P06241 8/20 0.48
PIK3CA P42336 9/20 0.46
HASPIN Q8TF76 2/20 0.42
KCNH2 Q12809 2/20 0.42
KIT P10721 1/20 0.42
PIM1 P11309 1/20 0.42
FLT3 P36888 1/20 0.42
CDK7 P50613 1/20 0.42
PIM3 Q86V86 1/20 0.42
PIM2 Q9P1W9 1/20 0.42
DPP4 P27487 1/20 0.40
DPP7 Q9UHL4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627458 1.00 FYN (0.48) FYNPIK3CAHASPINKCNH2KIT
SCHEMBL628259 0.87 DPP4 (0.38) FYNPIK3CAKCNH2DPP4DPP7
SCHEMBL628257 0.87 DPP4 (0.38) FYNPIK3CAKCNH2DPP4DPP7
SCHEMBL628258 0.87 DPP4 (0.38) FYNPIK3CAKCNH2DPP4DPP7
SCHEMBL627457 0.86 DPP4 (0.40) FYNPIK3CAKCNH2DPP4DPP7
SCHEMBL627441 0.81 FYN (0.63) FYNPIK3CAHASPIN
SCHEMBL627439 0.81 FYN (0.63) FYNPIK3CAHASPIN
SCHEMBL625300 0.80 PIK3CA (0.51) FYNPIK3CAHASPIN
SCHEMBL626206 0.80 PIK3CA (0.53) FYNPIK3CAHASPIN
SCHEMBL627396 0.79 PIK3CA (0.53) FYNPIK3CAHASPIN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed