SCHEMBL627457

SCHEMBL627457

Nc1ncc(-c2cn3nc(NC4CCC(NS(=O)(=O)c5ccc(F)cc5F)CC4)sc3n2)cc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 7/20 0.40
DPP7 Q9UHL4 5/20 0.40
KCNH2 Q12809 4/20 0.39
PIK3CA P42336 2/20 0.38
DPP8 Q6V1X1 3/20 0.38
DPP9 Q86TI2 3/20 0.38
MAP3K12 Q12852 6/20 0.38
F2RL3 Q96RI0 1/20 0.36
TNF P01375 1/20 0.36
ALOX5AP P20292 2/20 0.35
FEN1 P39748 2/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
FYN P06241 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627456 0.86 FYN (0.48) DPP4DPP7KCNH2PIK3CAFYN
SCHEMBL627458 0.86 FYN (0.48) DPP4DPP7KCNH2PIK3CAFYN
SCHEMBL628259 0.84 DPP4 (0.38) DPP4DPP7KCNH2PIK3CADPP8
SCHEMBL628257 0.84 DPP4 (0.38) DPP4DPP7KCNH2PIK3CADPP8
SCHEMBL628258 0.84 DPP4 (0.38) DPP4DPP7KCNH2PIK3CADPP8
SCHEMBL627440 0.81 FYN (0.45) PIK3CAMAP3K12FYN
SCHEMBL625301 0.80 MAP3K12 (0.44) PIK3CAMAP3K12PIK3CDPIK3CBPIK3CG
SCHEMBL626207 0.80 MAP3K12 (0.46) PIK3CAMAP3K12
SCHEMBL627397 0.80 PIK3CA (0.49) PIK3CAMAP3K12PIK3CDPIK3CBPIK3CG
SCHEMBL625236 0.80 MAP3K12 (0.45) PIK3CAMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed