SCHEMBL6274944

SCHEMBL6274944

O=C1[N]NN(c2cccc(Cl)c2)N1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 5/20 0.45
MGLL Q99685 1/20 0.44
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
TP53 P04637 1/20 0.41
ADRB1 P08588 1/20 0.41
CYP3A4 P08684 1/20 0.41
HTR1A P08908 1/20 0.41
CYP2D6 P10635 1/20 0.41
THRB P10828 1/20 0.41
CYP2C9 P11712 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
SLC6A4 P31645 1/20 0.41
HTR7 P34969 1/20 0.41
HTR2B P41595 1/20 0.41
HTT P42858 1/20 0.41
HTR3A P46098 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6270872 0.81 ALDH1A1 (0.46) ALOX5MGLLHTR2AHTR2CHTR2B
SCHEMBL1827924 0.78 HTT (0.51) ALOX5CYP1A2HTR3EHTR3BTHRB
SCHEMBL16296350 0.70 ALOX5 (0.47) ALOX5MGLLCYP1A2CYP2C19HTR3E
SCHEMBL6272012 0.69 S100A9 (0.40) NOTUM
SCHEMBL6273466 0.69 DAO (0.49) CYP2C19CYP2C9HTR2CMAPTHPGD
SCHEMBL2963118 0.67 MAPT (0.44) CYP1A2CYP2C9HTTMAPTGAA
SCHEMBL10948802 0.66 MEN1 (0.49) ALOX5MGLLCYP1A2CYP2C19HTR3E
SCHEMBL9623886 0.65 ALDH1A1 (0.71) ALOX5MGLLCYP1A2CYP2C19HTR3E
SCHEMBL2541490 0.65 IDO1 (0.60) MGLLCYP1A2CYP2C19HTR3EHTR3B
SCHEMBL3013325 0.64 GAA (0.59) ALOX5MGLLCYP1A2CYP2C19HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3008055-A1 NOVEL TETRAZOLONE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2016-04-20 EP disclosed
WO-2014198592-A1 NOVEL TETRAZOLONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2014-12-18 WO disclosed
EP-1606271-A1 INSECTICIDAL PHTHALAMIDE DERIVATIVES Bayer CropScience AG (DE) 2005-12-21 EP disclosed
WO-2004080984-A1 INSECTICIDAL PHTHALAMIDE DERIVATIVES BAYER CROPSCIENCE AG (DE) 2004-09-23 WO disclosed