SCHEMBL6277448

SCHEMBL6277448

O=[N+]([O-])c1c(Cl)ccnc1NCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.60
CA1 P00915 3/20 0.55
CA2 P00918 3/20 0.55
CA7 P43166 3/20 0.55
CA13 Q8N1Q1 3/20 0.55
MAPT P10636 5/20 0.53
KDM4E B2RXH2 1/20 0.50
LMNA P02545 3/20 0.49
MAPK1 P28482 2/20 0.49
HPGD P15428 1/20 0.49
ALDH1A1 P00352 2/20 0.48
EGFR P00533 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
POLB P06746 2/20 0.47
NPC1 O15118 2/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28068214 0.86 MAPT (0.62) HTTCA1CA2CA7CA13
SCHEMBL4743191 0.84 HTT (0.61) HTTCA1CA2CA7CA13
SCHEMBL8562625 0.83 HTT (0.67) HTTCA1CA2CA7CA13
SCHEMBL30983973 0.81 HTT (0.71) HTTCA1CA2CA7CA13
SCHEMBL18359454 0.80 PGK1 (0.48) HTTMAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL16345563 0.78 PIN1 (0.52) HTTCA1CA2CA7CA13
SCHEMBL2572082 0.78 HTT (0.50) HTTCA1CA2CA7CA13
SCHEMBL5033956 0.76 HTT (0.52) HTTCA1CA2CA7CA13
SCHEMBL31631301 0.75 NPC1 (0.74) HTTCA1CA2CA7CA13
SCHEMBL1738419 0.75 NPC1 (0.74) HTTCA1CA2CA7CA13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005121094-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES AS ANTI-HIV-AGENTS PFIZER LIMITED (GB) 2005-12-22 WO disclosed