SCHEMBL6278367

SCHEMBL6278367

O=C(CCN1CCCCC1)Nc1cc[c]cc1

nearest known ligand 0.73

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.73
POLB P06746 1/20 0.73
KMT2A Q03164 2/20 0.68
LMNA P02545 2/20 0.68
MEN1 O00255 1/20 0.68
MAPT P10636 2/20 0.64
ALOX15 P16050 1/20 0.64
GLA P06280 1/20 0.61
ATM Q13315 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
TSHR P16473 1/20 0.61
MAPK1 P28482 1/20 0.60
TERT O14746 6/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1355051 0.98 ALDH1A1 (0.70) ALDH1A1POLBKMT2ALMNAMEN1
SCHEMBL1356631 0.87 TP53 (0.70) ALDH1A1LMNAMAPTTERT
SCHEMBL962893 0.85 LMNA (0.74) ALDH1A1POLBKMT2ALMNAALOX15
SCHEMBL2180527 0.85 LMNA (0.54) ALDH1A1POLBKMT2ALMNAMEN1
SCHEMBL3012622 0.84 ALDH1A1 (1.00) ALDH1A1POLBKMT2ALMNAMEN1
SCHEMBL22407734 0.84 KDM4E (0.68) ALDH1A1POLBKMT2ALMNAMEN1
SCHEMBL1355900 0.84 KDM4E (0.68) ALDH1A1POLBKMT2ALMNAMEN1
SCHEMBL6492893 0.83 LMNA (0.56) ALDH1A1POLBKMT2ALMNAMEN1
SCHEMBL1355565 0.83 KDM4E (0.67) ALDH1A1POLBKMT2ALMNAMEN1
SCHEMBL13149726 0.82 KMT2A (0.97) ALDH1A1POLBKMT2ALMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836613-B1 WATER-SOLUBLE ADENOSINE KINASE INHIBITORS METABASIS THERAPEUTICS INC (US) 2005-05-25 EP disclosed
US-5795977-A Water soluble adenosine kinase inhibitors METABASIS THERAPEUTICS, INC. (US) 1998-08-18 US disclosed
EP-0836613-A1 WATER-SOLUBLE ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-22 EP disclosed
US-5726302-A SUBSTITUTED 4-AMINO PYRROLO(2,3-D) PYRIMIDINE AND PYRAZOLO(3,4-D) PYRIMIDINE NUCLEOSIDE ANALOGS GENSIA INC. (US) 1998-03-10 US disclosed
WO-1996040707-A1 WATER-SOLUBLE ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed