SCHEMBL6281696

SCHEMBL6281696

CC(C)(C)NC(=O)[C@@H]1CC[C@H](CO)N1C(=O)OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.46
FKBP1A P62942 2/20 0.44
HTT P42858 1/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
AGTR2 P50052 1/20 0.43
NPSR1 Q6W5P4 2/20 0.42
TSHR P16473 2/20 0.42
KDM4E B2RXH2 2/20 0.42
LMNA P02545 2/20 0.42
TP53 P04637 1/20 0.42
GLA P06280 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
THPO P40225 1/20 0.42
HIF1A Q16665 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6286208 0.85 HTT (0.42) HTR2CFKBP1AHTTNPC1RAB9A
SCHEMBL6278076 0.85 HTR2C (0.41) HTR2CFKBP1AHTTNPC1RAB9A
SCHEMBL9546482 0.83 SMN1; SMN2 (0.52) HTR2CNPC1RAB9ASMN1; SMN2AGTR2
SCHEMBL9546475 0.83 SMN1; SMN2 (0.52) HTR2CNPC1RAB9ASMN1; SMN2AGTR2
SCHEMBL7376563 0.83 HTR2C (0.47) HTR2CFKBP1AHTTNPC1RAB9A
SCHEMBL9546620 0.82 HTR2C (0.57) HTR2CNPC1RAB9ASMN1; SMN2AGTR2
SCHEMBL18410564 0.82 HTR2C (0.57) HTR2CNPC1RAB9ASMN1; SMN2AGTR2
SCHEMBL13958801 0.78 NPSR1 (0.66) RAB9ANPSR1TSHRKDM4ELMNA
SCHEMBL28411856 0.76 HTR2C (0.47) HTR2CHTTNPC1RAB9ASMN1; SMN2
SCHEMBL28414267 0.76 HTR2C (0.52) HTR2CHTTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6900238-B1 HIV protease inhibitors THE SCRIPPS RESEARCH INSTITUTE (US) 2005-05-31 US disclosed
EP-0873519-A4 HIV PROTEASE INHIBITORS SCRIPPS RESEARCH INST (US) 2005-04-27 EP disclosed
EP-0873519-A1 HIV PROTEASE INHIBITORS The Scripps Research Institute (US) 1998-10-28 EP disclosed
WO-1997021100-A9 HIV PROTEASE INHIBITORS 1997-10-30 WO disclosed
WO-1997021100-A1 HIV PROTEASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 1997-06-12 WO disclosed