SCHEMBL6286208

SCHEMBL6286208

CCCC(=O)OC[C@H]1CC[C@@H](C(=O)NC(C)(C)C)N1C(=O)OCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
PRCP P42785 1/20 0.41
HTR2C P28335 1/20 0.41
TSHR P16473 2/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TP53 P04637 1/20 0.41
GLA P06280 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
THPO P40225 1/20 0.41
HIF1A Q16665 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GMNN O75496 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6282539 0.87 HTR2C (0.46) HTTPRCPHTR2CSMN1; SMN2NPC1
SCHEMBL6281696 0.85 HTR2C (0.46) HTTHTR2CTSHRKDM4ELMNA
SCHEMBL6278076 0.83 HTR2C (0.41) HTTHTR2CTSHRKDM4ELMNA
SCHEMBL28411856 0.75 HTR2C (0.47) HTTPRCPHTR2CTSHRKDM4E
SCHEMBL13958801 0.73 NPSR1 (0.66) PRCPTSHRKDM4ELMNANPSR1
SCHEMBL1509090 0.72 HTR2C (0.53) HTTHTR2CNPSR1ALDH1A1SMN1; SMN2
SCHEMBL13567880 0.72 HTR2C (0.53) HTTHTR2CNPSR1ALDH1A1SMN1; SMN2
SCHEMBL29816886 0.72 HTR2C (0.48) HTTPRCPHTR2CTSHRKDM4E
SCHEMBL29816690 0.72 HTR2C (0.48) HTTPRCPHTR2CTSHRKDM4E
SCHEMBL29816802 0.72 HTR2C (0.48) HTTPRCPHTR2CTSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6900238-B1 HIV protease inhibitors THE SCRIPPS RESEARCH INSTITUTE (US) 2005-05-31 US disclosed
EP-0873519-A4 HIV PROTEASE INHIBITORS SCRIPPS RESEARCH INST (US) 2005-04-27 EP disclosed
EP-0873519-A1 HIV PROTEASE INHIBITORS The Scripps Research Institute (US) 1998-10-28 EP disclosed
WO-1997021100-A9 HIV PROTEASE INHIBITORS 1997-10-30 WO disclosed
WO-1997021100-A1 HIV PROTEASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 1997-06-12 WO disclosed