SCHEMBL6278076

SCHEMBL6278076

CC(C)(C)NC(=O)[C@@H]1CC[C@H](CO[Si](C)(C)C(C)(C)C)N1C(=O)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.41
NPSR1 Q6W5P4 2/20 0.41
TSHR P16473 2/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
HSD17B10 Q99714 2/20 0.41
TP53 P04637 1/20 0.41
GLA P06280 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
THPO P40225 1/20 0.41
HIF1A Q16665 1/20 0.41
GMNN O75496 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
MTOR P42345 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6281696 0.85 HTR2C (0.46) HTR2CNPSR1TSHRKDM4ELMNA
SCHEMBL6286208 0.83 HTT (0.42) HTR2CNPSR1TSHRKDM4ELMNA
SCHEMBL29560191 0.77 SMN1; SMN2 (0.45) NPC1RAB9ASMN1; SMN2PREP
SCHEMBL30781570 0.76 POLB (0.44) HTR2CNPC1RAB9ASMN1; SMN2AGTR2
SCHEMBL6475389 0.76 PREP (0.49) NPSR1TSHRKDM4ELMNAHSD17B10
SCHEMBL6475398 0.76 PREP (0.49) NPSR1TSHRKDM4ELMNAHSD17B10
SCHEMBL6484219 0.76 PREP (0.49) NPSR1TSHRKDM4ELMNAHSD17B10
SCHEMBL31390598 0.75 CTSL (0.41) HTR2CHPGDFKBP1ASMN1; SMN2L3MBTL1
SCHEMBL2727664 0.75 SMN1; SMN2 (0.41) HTR2CNPSR1NPC1RAB9ASMN1; SMN2
SCHEMBL2843333 0.75 SMN1; SMN2 (0.41) HTR2CNPSR1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6900238-B1 HIV protease inhibitors THE SCRIPPS RESEARCH INSTITUTE (US) 2005-05-31 US disclosed
WO-1997021100-A9 HIV PROTEASE INHIBITORS 1997-10-30 WO disclosed