SCHEMBL6282047

SCHEMBL6282047

COCOc1ccc(-c2cccc3c2c(/C=C/c2ccccc2)nn3COCC[Si](C)(C)C)cc1OC

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.34
EGFR P00533 1/20 0.34
IGF1R P08069 1/20 0.34
SRC P12931 1/20 0.34
FLT4 P35916 1/20 0.34
FLT3 P36888 1/20 0.34
EPHB4 P54760 1/20 0.34
TEK Q02763 1/20 0.34
GAK O14976 1/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP1B1 Q16678 1/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 2/20 0.32
HSD17B10 Q99714 2/20 0.32
ALDH1A1 P00352 2/20 0.32
NPC1 O15118 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6282051 1.00 KDR (0.34) KDREGFRIGF1RSRCFLT4
SCHEMBL5250921 0.85 KDR (0.36) KDREGFRIGF1RSRCFLT4
SCHEMBL5250919 0.85 KDR (0.36) KDREGFRIGF1RSRCFLT4
SCHEMBL14493402 0.77 EGFR (0.34) KDREGFRIGF1RSRCFLT4
SCHEMBL6283631 0.76 RET (0.35) RAB9AKDM4EALDH1A1NPC1HPGD
SCHEMBL6283634 0.76 RET (0.35) RAB9AKDM4EALDH1A1NPC1HPGD
SCHEMBL5246902 0.74 PTGS2 (0.42) RAB9AKDM4EALDH1A1NPC1GAA
SCHEMBL5246898 0.74 PTGS2 (0.42) RAB9AKDM4EALDH1A1NPC1GAA
SCHEMBL5526396 0.70 CHEK1 (0.39) KDREGFRNPC1
SCHEMBL14493368 0.70 CHEK1 (0.39) KDREGFRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6891044-B2 Indazole compounds and pharmaceutical compositions for Inhibiting protein kinases, and methods for their use AGOURON PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed