SCHEMBL6283631

SCHEMBL6283631

C[Si](C)(C)CCOCn1nc(/C=C/c2ccccc2)c2c(N)cccc21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.35
NPC1 O15118 5/20 0.33
KDM4E B2RXH2 4/20 0.32
ALDH1A1 P00352 4/20 0.32
RAB9A P51151 4/20 0.32
SMN1; SMN2 Q16637 4/20 0.32
PKM P14618 2/20 0.32
NFKB1 P19838 2/20 0.32
NFKB2 Q00653 2/20 0.32
RELA Q04206 2/20 0.32
GAA P10253 3/20 0.32
GLA P06280 2/20 0.32
MAPT P10636 2/20 0.32
HPGD P15428 2/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
GRM4 Q14833 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6283634 1.00 RET (0.35) RETNPC1KDM4EALDH1A1RAB9A
SCHEMBL6285089 0.82 F2RL1 (0.34) RETNPC1
SCHEMBL27615251 0.80 CNR1 (0.37) RETNPC1KDM4EALDH1A1MAPT
SCHEMBL5248918 0.80 KDR (0.35) RETNPC1GRM4ALOX5APFEN1
SCHEMBL5248919 0.80 KDR (0.35) RETNPC1GRM4ALOX5APFEN1
SCHEMBL25170244 0.78 ALOX5AP (0.35) NPC1ALOX5APFEN1
SCHEMBL5512063 0.78 NPC1 (0.36) NPC1KDM4EALDH1A1RAB9ASMN1; SMN2
SCHEMBL7511036 0.78 NPC1 (0.36) NPC1KDM4EALDH1A1RAB9ASMN1; SMN2
SCHEMBL5514694 0.77 NPC1 (0.33) NPC1ALOX5APFEN1
SCHEMBL7507059 0.77 NPC1 (0.33) NPC1ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6891044-B2 Indazole compounds and pharmaceutical compositions for Inhibiting protein kinases, and methods for their use AGOURON PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed