SCHEMBL628244

SCHEMBL628244

Ic1cn2nc(NC3CCOCC3)sc2n1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.36
PDE10A Q9Y233 2/20 0.35
FYN P06241 4/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
MKNK1 Q9BUB5 2/20 0.32
CCNE1 P24864 4/20 0.31
CDK2 P24941 4/20 0.31
MKNK2 Q9HBH9 1/20 0.31
CNR2 P34972 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE7A Q13946 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625118 0.84 POLB (0.31) MAPK1
SCHEMBL627168 0.78 CCNE1 (0.39) CCNE1CDK2
SCHEMBL626399 0.74 KDM1A (0.38) CDK2
SCHEMBL2254823 0.74 EGLN1 (0.40) CNR2
SCHEMBL627884 0.74 CCNA2 (0.50) MAPK1CDK2
SCHEMBL628243 0.73 FYN (0.46) MAPK1FYNMKNK1
SCHEMBL2255826 0.72 FYN (0.52) FYNPDE4B
SCHEMBL2252684 0.72 F2RL3 (0.40) MAPK1PDE10A
SCHEMBL625292 0.69 PIM1 (0.53)
SCHEMBL624035 0.69 SMN1; SMN2 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed