SCHEMBL627168

SCHEMBL627168

CS(=O)(=O)N1CCC(Nc2nn3cc(I)nc3s2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 16/20 0.39
CDK2 P24941 16/20 0.39
CCNE2 O96020 4/20 0.39
CCNB2 O95067 3/20 0.39
CDK1 P06493 3/20 0.39
CCNB1 P14635 3/20 0.39
CDK5 Q00535 3/20 0.39
CDK5R1 Q15078 3/20 0.39
CCNB3 Q8WWL7 3/20 0.39
CCND1 P24385 6/20 0.39
CDK6 Q00534 6/20 0.39
CCNT1 O60563 5/20 0.39
CDK4 P11802 5/20 0.39
CDK9 P50750 5/20 0.39
IKBKB O14920 1/20 0.38
JAK2 O60674 1/20 0.37
JAK3 P52333 1/20 0.37
PTK2 Q05397 1/20 0.37
IDO1 P14902 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627200 0.84 POLB (0.35) CDK2IKBKB
SCHEMBL628244 0.78 MAPK1 (0.36) CCNE1CDK2
SCHEMBL626172 0.78 DYRK1A (0.38) CCNE1CDK2CCNE2CCNB2CDK1
SCHEMBL627884 0.77 CCNA2 (0.50) CDK2
SCHEMBL627492 0.77 CDK2 (0.39) CCNE1CDK2CCNE2CCNB2CDK1
SCHEMBL627167 0.77 FYN (0.46) CCNE1CDK2CCNE2CCNB2CDK1
SCHEMBL627493 0.77 CCNE1 (0.37) CCNE1CDK2CCNE2CCNB2CDK1
SCHEMBL624133 0.77 RORC (0.34) JAK2IDO1
SCHEMBL627850 0.76 JAK1 (0.35) CDK2JAK3
SCHEMBL623928 0.76 FYN (0.49) CDK2CDK1CDK5CCND1CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed