SCHEMBL628253

SCHEMBL628253

OC1CCC(CNc2nn3cc(I)nc3s2)CC1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.40
FYN P06241 8/20 0.39
PI4KB Q9UBF8 2/20 0.33
PDE10A Q9Y233 1/20 0.32
PIK3CA P42336 1/20 0.32
PI4KA P42356 1/20 0.32
PIK3CG P48736 1/20 0.32
VNN1 O95497 1/20 0.32
IRAK1 P51617 1/20 0.31
GRIN2B Q13224 1/20 0.31
PIM1 P11309 1/20 0.31
NPY5R Q15761 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2257064 0.94 MKNK1 (0.44) MKNK1FYNPI4KBPDE10APIK3CA
SCHEMBL627315 0.84 MKNK1 (0.37) MKNK1FYNVNN1NPY5R
SCHEMBL627067 0.78 KDM4E (0.46) GRIN2BNPY5R
SCHEMBL15324843 0.77 MKNK1 (0.42) MKNK1FYNPI4KBPDE10APIK3CA
SCHEMBL628252 0.75 MKNK1 (0.57) MKNK1FYNVNN1PIM1
SCHEMBL628254 0.75 MKNK1 (0.57) MKNK1FYNVNN1PIM1
SCHEMBL1944318 0.74 MKNK1 (0.45) MKNK1FYN
SCHEMBL1944253 0.72 TP53 (0.53) MKNK1FYN
SCHEMBL1945276 0.72 MAPT (0.45) MKNK1FYN
SCHEMBL627611 0.72 MAP3K12 (0.43) FYNPIK3CAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed