SCHEMBL6282874

SCHEMBL6282874

N#Cc1ccc(OCc2ccccc2)c(C2Cc3ccccc3N(CCCCCBr)C2=O)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.39
KCNH2 Q12809 3/20 0.39
PTGER1 P34995 1/20 0.36
MAOB P27338 1/20 0.36
TDP2 O95551 2/20 0.36
MRGPRX4 Q96LA9 3/20 0.36
SLC6A9 P48067 1/20 0.35
HDAC6 Q9UBN7 3/20 0.35
MET P08581 2/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
CDK2 P24941 1/20 0.34
CDK9 P50750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7119871 0.83 F10 (0.39) MRGPRX4
SCHEMBL7124449 0.83 F10 (0.39) MRGPRX4
SCHEMBL6280175 0.79 HTR7 (0.37) KCNH2DRD2DRD4DRD3
SCHEMBL6275380 0.75 MAOB (0.42) HTR6KCNH2PTGER1MAOBTDP2
SCHEMBL7116050 0.74 F10 (0.39)
SCHEMBL7413976 0.72 TNKS2 (0.43) HTR6PTGER1MAOBTDP2MRGPRX4
SCHEMBL7126646 0.72 F10 (0.59)
SCHEMBL7121499 0.72 F10 (0.59)
SCHEMBL6278778 0.72 F10 (0.53) HDAC6
SCHEMBL6281661 0.68 CACNA1S (0.53) HDAC6DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6855726-B1 Quinolones as serine protease inhibitors WARNER-LAMBERT COMPANY LLC (US) 2005-02-15 US disclosed
EP-1091955-A1 QUINOLONES AS SERINE PROTEASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2001-04-18 EP disclosed
WO-1999050263-A1 QUINOLONES AS SERINE PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1999-10-07 WO disclosed